Qoraa: Gregory Harris
Taariikhda Abuurista: 8 Abriil 2021
Taariikhda Cusboonaysiinta: 15 Laga Yaabaa 2024
Anonim
Linezolid (Oxazolidinone Antibiotic) - Mechanism of Action, Indications, and Side Effects
Dareemoleyad: Linezolid (Oxazolidinone Antibiotic) - Mechanism of Action, Indications, and Side Effects

Qanacsan

Linezolid waxaa loo isticmaalaa in lagu daaweeyo infekshannada, oo ay kujiraan oofwareenka, iyo infekshannada maqaarka. Linezolid waxay kujirtaa fasal lidka bakteeriyada loo yaqaan oxazolidinones. Waxay ku shaqeysaa joojinta koritaanka bakteeriyada.

Antibiyootikada sida linezolid uma shaqeyn doonto hargabka, ifilada, iyo infekshannada kale ee fayraska ku dhaca. Isticmaalka antibiyootikada markii aan loo baahnayn waxay kordhisaa halista aad u qaadi karto jeermis dambe oo iska caabiya daaweynta antibiyootikada.

Linezolid waxay u timaadaa sidii kaniiniga iyo ka joojinta afka (dareeraha) si afka looga qaato. Waxaa badanaa la qaataa ama cunno la'aan laba jeer maalintii (12-kii saacadoodba) 10 ilaa 28 maalmood. Carruurta da'doodu tahay 11 sano iyo wixii ka yar sida caadiga ah waxay qaataan 'linezolid' ama cunno la'aan laba ilaa saddex jeer maalintii (8 ilaa 12 saacadood kasta) 10 illaa 28 maalmood. Dhererka daaweyntaadu waxay kuxirantahay nooca cudurka aad qabtid. Si taxaddar leh u raac tilmaamaha ku qoran calaamadaha laguu qoray, oo weydii takhtarkaaga ama farmashiistaha inuu kuu sharxo qayb kasta oo aadan fahmin. Qaado linezolid sida saxda ah ee lagu faray. Ha ka qaadin wax ka yar ama ka yar ama u qaado si ka badan inta dhakhtarku kuu qoray.


Kahor intaadan isticmaalin ka joojinta afka, si tartiib ah isku qas adigoo dhalada isku rogaya seddex ilaa shan jeer. Ha ruxin ganaaxa.

Qaado dawada loo yaqaan 'linezolid' illaa aad ka dhammeysid rijeetada laguu qoray, xitaa haddii aad fiicnaan dareento. Ha u joojin qaadashada daawada 'linezolid' adiga oo aan la hadlin dhakhtarkaaga. Haddii aad joojiso qaadashada daawada 'linezolid' dhaqso ama haddii aad ka boodo qiyaasaha, cudurkaaga waxaa laga yaabaa in aan gebi ahaanba la daaweyn oo ay bakteeriyadu u adkeysato antibiyootikada

Daawadan waxaa loo qori karaa adeegsiyo kale; Weydii dhakhtarkaaga ama farmashiistaha wixii macluumaad dheeraad ah.

Kahor qaadashada linezolid,

  • u sheeg dhakhtarkaaga iyo farmashiistahaaga haddii aad xasaasiyad ku leedahay linezolid, daawooyinka kale, ama mid ka mid ah waxyaabaha ku jira sheyga linezolid ee laguu qoray. Weydii farmashiistahaaga liiska waxyaabaha ay ka kooban yihiin.
  • u sheeg dhakhtarkaaga haddii aad qaadanaysid dawooyinka soo socda ama aad joojisay qaadashadooda labadii toddobaad ee la soo dhaafay: isocarboxazid (Marplan) phenelzine (Nardil). rasagiline (Azilect), selegiline (Eldepryl, Emsam, Zelapar), iyo tranylcypromine (Parnate). Dhakhtarkaaga ayaa laga yaabaa inuu kuu sheego inaadan qaadan linezolid haddii aad qaadanaysid mid ama in kabadan oo daawooyinkan ah, ama aad qaadatay labadii todobaad ee lasoo dhaafay.
  • u sheeg dhakhtarkaaga iyo farmashiistaha waxa kale ee dhakhtar qoro iyo kuwa aan dhakhtar qorin, fiitamiinnada, nafaqada nafaqada, iyo alaabta dhirta ah ee aad qaadanayso ama aad qorsheyneyso inaad qaadato. Hubso inaad sheegto mid ka mid ah kuwan soo socda: epinephrine (EpiPen); meperidine (Demerol); dawooyinka dhanjafka sida almotriptan (Axert), eletriptan (Relpax), frovatriptan (Frova), naratriptan (Amerge), rizatriptan (Maxalt), sumatriptan (Imitrex, in Treximet), iyo zolmitriptan (Zomig); phenylpropanolamine (oo aan hadda laga heli karin Maraykanka); iyo pseudoephedrine (Sudafed; dawooyin badan oo qabow ama sunta baabi'isa). Sidoo kale u sheeg dhakhtarkaaga haddii aad qaadanaysid daawooyinka soo socda ama aad joojisay qaadashadooda labadii toddobaad ee la soo dhaafay: bupropion (Aplenzin, Wellbutrin, Zyban, kuwo kale); buspirone; xulashada serotonin reuptake inhibitors (SSRIs) sida citalopram (Celexa), escitalopram (Lexapro), fluvoxamine (Luvox), paroxetine (Brisdelle, Paxil, Pexeva), sertraline (Zoloft), iyo vilazodone (Vilbyrd); serotonin norepinephrine reuptake inhibitors (SNRIs) sida desvenlafaxine (Khedezla, Pristiq), duloxetine (Cymbalta), levomilnacipran (Fetzima), iyo venlafaxine (Effexor); iyo daawada murugada ee tricyclic sida amitriptyline, amoxapine, clomipramine (Anafranil), desipramine (Norpramin), doxepin (Silenor), imipramine (Tofranil), nortriptyline (Pamelor), protriptyline (Vivactil), iyo trimipramine (Sur) Sidoo kale u sheeg dhakhtarkaaga haddii aad qaadanayso fluoxetine (Prozac, Sarafem, Selfemra, oo ku taal Symbyax), ama aad joojisay qaadashadiisa 5tii toddobaad ee la soo dhaafay. Dhakhtarkaaga ayaa laga yaabaa inuu u baahdo inuu beddelo qiyaasta daawooyinkaaga ama uu si taxaddar leh kuugu ilaaliyo dhibaatooyinka soo raaca. Daawooyin kale oo badan ayaa sidoo kale la macaamili kara linezolid, markaa hubi inaad u sheegto dhakhtarkaaga dhammaan daawooyinka aad qaadanaysid, xitaa kuwa aan ka muuqan liiskan.
  • u sheeg dhakhtarkaaga haddii aad qabtid infakshan daba-dheeraada (muddo dheer soconaya), ama haddii aad leedahay ama aad waligaa yeelatay cudurka kansarka (xaalad buro ku soo saarto serotonin). sonkorowga, dhiig karka, hyperthyroidism (qanjirka 'thyroid'), xakamaynta difaaca jirka (dhibaatooyinka nidaamkaaga difaaca), pheochromocytoma (buro ku taal qanjirka 'adrenal gland'), qalal, ama cudur kalyaha ah.
  • u sheeg dhakhtarkaaga haddii aad uur leedahay, qorsheyso inaad uur yeelato, ama aad naas nuujiso. Haddii aad uur yeelato inta aad qaadanaysid daawada loo yaqaan 'linezolid', wac dhakhtarkaaga.
  • haddii aad qalliin samaynayso, oo ay ku jiraan qalliinka ilkaha, u sheeg dhakhtarka ama dhakhtarka ilkaha in aad qaadanayso dawada loo yaqaan 'linezolid'.
  • haddii aad leedahay phenylketonuria (PKU, xaalad la iska dhaxlo oo ah in cunno gaar ah la raaco si looga hortago dib-u-dhac maskaxeed), waa inaad ogaataa in joojinta afka ay kujirto aspartame oo sameysa phenylalanine.

Ka fogow cunista ama cabidda tiro badan oo ah cuntooyin iyo cabitaanno ay ku jiraan maadada 'tyramine' inta aad qaadaneysid daawada loo yaqaan 'linezolid'. Cunnooyinka iyo cabbitaannada la kariyey, la qiijiyey, ama la khamiiryey badiyaa waxay ku jiraan maaddada 'tyramine'. Cuntooyinkan iyo cabitaannadan waxaa ka mid ah cabbitaannada aalkolada ah, gaar ahaan biirka, Chianti, iyo khamri kale oo cas; biir aan khamri lahayn; jiis (gaar ahaan xoog badan, da 'weyn, ama noocyo la farsameeyay); sauerkraut; yogurt; sabiib; muuska; labeen dhanaan; herring pickled; beerka (gaar ahaan beerka digaagga); Hilib iyo bolse qalalan (oo ay ku jiraan salami adag iyo basbaas); berde qasacadaysan; avocados; maraqa soy; turkey; soosaarida khamiirka; waxsoosaarka babayga (oo ay kujiraan jilciyayaal hilib qaarkood); digirta fava; iyo qeybaha digirta ballaaran.


Qaado qiyaasta la seegay isla marka aad xasuusatoba. Si kastaba ha noqotee, haddii ay ku dhowdahay waqtiga qiyaasta xigta, ka bood qiyaasta la seegay oo sii wad jadwalka daawadaada caadiga ah. Ha qaadan laba-qaadasho si aad uhesho mid kaa dhaafay.

Linezolid waxay sababi kartaa waxyeelo. U sheeg dhakhtarkaaga haddii mid ka mid ah astaamahani ay daran yihiin ama aanad tagin:

  • shuban
  • madax xanuun
  • lallabbo
  • matagid
  • calool xanuun
  • beddel sida ay wax u dhadhamiyaan
  • finan
  • cuncun
  • dawakhaad
  • balastarro cadcad oo afka ah
  • cuncun, gubasho, ama cuncun siilka
  • midabka carrabka ama ilkaha oo is beddela

Dhibaatooyinka qaarkood waxay noqon karaan kuwo halis ah. Haddii aad isku aragto mid ka mid ah astaamahan, wac takhtarkaaga isla markiiba ama u hesho daaweyn caafimaad oo deg-deg ah:

  • cuncun, finan, cuncun, neefsashada ama wax liqidda oo ku adkaata, barar wejiga, cunaha, carrabka, bushimaha, indhaha, gacmaha, cagaha, anqawyada, ama lugaha hoose, xabeeb
  • maqaarka oo bararaya ama fiiqan
  • lallabbo iyo matag soo noqnoqday; neefsashada degdegga ah; jahwareer; daal dareemid
  • xanuun, kabuubyo, ama daciifnimo gacmaha, cagaha, ama qaybaha kale ee jirka
  • shuban daran (saxaro biyo ah ama dhiig leh) oo ku dhici kara xummad ama aan lahayn iyo calool xanuun (waxay dhici kartaa ilaa 2 bilood ama ka badan daaweyntaada ka dib)
  • dhiigbax ama nabar aan caadi ahayn
  • isbeddelada aragtida midabka, aragga daciifka ah, ama isbeddelada kale ee aragga
  • qalal

Linezolid waxay sababi kartaa waxyeelo kale. Wac dhakhtarkaaga haddii aad qabtid dhibaatooyin aan caadi ahayn intaad qaadanaysid dawadan.


Haddii aad isku aragto waxyeellooyin daran, adiga ama dhakhtarkaaga ayaa warbixin u diri kara Barnaamijka Ka Warbixinta Dhacdooyinka Xun ee Maamulka Cuntada iyo Dawooyinka (FDA) (http://www.fda.gov/Safety/MedWatch) ama taleefan ( 1-800-332-1088).

Daawadan ku hay weelka ay soo gashay, si adag u xir, iyo meel aysan carruurtu gaarin. Ku keydi heerkulka qolka oo ka fog iftiinka iyo kuleylka badan iyo qoyaanka (ha ku jirin musqusha). Hakinta afka Linezolid waa in lagu isticmaalo 21 maalmood gudahood.

Daawooyinka aan loo baahnayn waa in lagu tuuraa siyaabo gaar ah si loo hubiyo in xayawaanka, carruurta, iyo dadka kaleba aysan cuni karin. Si kastaba ha noqotee, waa inaadan ku daadinin daawadan musqusha hoosteeda. Taabadalkeed, sida ugufiican ee dawada looga takhalusi karaa waa iyada oo loo maro barnaamijka dib u celinta daawada. La hadal farmashiistahaaga ama la xiriir waaxda qashinka / dib u warshadaynta si aad wax uga ogaato barnaamijyada dib-u-celinta ee bulshadaada. Ka eeg bogga internetka ee 'FDA ee Amni-Qaadashada Daawooyinka (http://goo.gl/c4Rm4p) si aad u hesho macluumaad dheeraad ah haddii aadan marin u helin barnaamijka dib-u-celinta.

Waa muhiim inaad ka ilaaliso dhammaan daawooyinka meel aan la arkeynin oo aysan gaari karin carruurta maaddaama weelal badan (sida kuwa toddobaadlaha kiniiniga ka fiirsada iyo kuwa loogu talagalay dhibcaha isha, kareemada, dhejiyeyaasha, iyo kuwa neefta ku siiya) uma adkeysana carruurta, carruurta yaryarna si fudud ayey ku furi karaan. Si aad uga ilaaliso carruurta yaryar sunta, marwalba xiro daboolka badbaadada isla markaana isla markiiba dhig dawada meel aamin ah - mid kor iyo fog kana fog aragooda oo gaadha. http://www.upandaway.org

Xaalada xad dhaafka ah, wac khadka caawinta ka hortagga sunta 1-800-222-1222. Macluumaadka sidoo kale waxaa laga heli karaa internetka https://www.poisonhelp.org/help.Haddii dhibbanuhu burburay, suuxdin qabtay, neefsashadu dhib ku tahay, ama aan la kici karin, isla markiiba wac adeegyada gurmadka ee 911.

Dhammaan ballamaha la dhig dhakhtarkaaga iyo shaybaarka. Dhakhtarkaaga ayaa laga yaabaa inuu amro baadhitaanada dhiigga qaarkood si loo hubiyo jawaabta jidhkaaga ee 'linezolid'.

Ha u ogolaan qof kale inuu qaato daawadaada. Takhtarka laguu qoray ayaa laga yaabaa inaan dib loo buuxin karin. Haddii aad wali leedahay calaamadaha cudurka ka dib markaad dhameysato linezolid, wac dhakhtarkaaga.

Waxaa muhiim kuu ah inaad haysato liis qoran oo ku saabsan dhammaan daawooyinka laguu qoro iyo kuwa aan dhakhtar qorin (warqad dhakhtar la aan ah) ee aad qaadanaysid, iyo sidoo kale wax soo saar kasta sida fiitamiinnada, macdanta, ama nafaqooyinka kale ee nafaqada leh. Waa inaad soo qaadataa liiskan markasta oo aad booqato dhakhtar ama haddii isbitaal la dhigo. Sidoo kale waa macluumaad muhiim ah inaad lasocoto haddii ay jiraan xaalado deg deg ah.

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